SCHEMBL7962995

SCHEMBL7962995

COc1cccc2c(CBr)coc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
HPGD P15428 3/20 0.49
LMNA P02545 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
PSMB8 P28062 1/20 0.46
PSMB5 P28074 1/20 0.46
HTR1A P08908 5/20 0.41
KDM4E B2RXH2 3/20 0.40
MAOA P21397 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
TBXA2R P21731 6/20 0.38
PTGIR P43119 6/20 0.38
GSK3B P49841 2/20 0.37
CDK2 P24941 1/20 0.37
MAPT P10636 2/20 0.36
CYP3A4 P08684 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CYP2A6 P11509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234354 0.87 ALDH1A1 (0.46) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL806348 0.85 ALDH1A1 (0.54) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL5761000 0.84 ALDH1A1 (0.48) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL7953106 0.83 ALDH1A1 (0.53) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL5763789 0.83 ALDH1A1 (0.47) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL4136821 0.81 MEN1 (0.46) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL4130976 0.81 PSMB8 (0.46) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL5504988 0.81 TAAR1 (0.53) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL21807593 0.80 PSMB5 (0.49) ALDH1A1HPGDLMNAMEN1KMT2A
SCHEMBL21807586 0.80 PSMB5 (0.44) ALDH1A1HPGDLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6323235-B1 CARDIOVASCULAR DISORDERS, ANTIISCHEMIC AGENTS AND ENZYME INHIBITORS OHTAKE ATSUSHI (JP) 2001-11-27 US disclosed
US-6043264-A A THROMBOXANE A2 RECEPTOR ANTAGONIST FOR TREATING HYPERTENSION, THROMBOSIS, ISCHEMIC HEART DISEASES, CIRCULATORY DISEASES, ARTERIOSCLEROSIS, PLATELET FUNCTION DISORDER, HYPERLIPIDEMIA, NEPHRITIS OR ASTHMA TORAY INDUSTRIES, INC. (JP) 2000-03-28 US disclosed
EP-0751126-A1 BENZENE-FUSED HETEROCYCLIC DERIVATIVE AND USE OF THE SAME TORAY INDUSTRIES, INC. (JP) 1997-01-02 EP disclosed