SCHEMBL7963333

SCHEMBL7963333

Cc1cccc2[nH]c(COc3cc(Cl)cc(Cl)c3)nc12

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 9/20 0.48
NPC1 O15118 8/20 0.48
SMN1; SMN2 Q16637 7/20 0.48
GAA P10253 6/20 0.48
MGAM O43451 5/20 0.48
SI P14410 5/20 0.48
MGAM2 Q2M2H8 5/20 0.48
POLB P06746 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
TP53 P04637 3/20 0.45
ALDH1A1 P00352 1/20 0.45
TSHR P16473 1/20 0.43
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7691472 0.91 GAA (0.53) RAB9ANPC1SMN1; SMN2GAAMGAM
SCHEMBL7689804 0.88 RAB9A (0.63) RAB9ANPC1SMN1; SMN2GAAMGAM
SCHEMBL7686239 0.84 GRIN1 (0.49) RAB9ANPC1SMN1; SMN2GAAPOLB
SCHEMBL8668275 0.83 RAB9A (0.61) RAB9ANPC1SMN1; SMN2GAAPOLB
SCHEMBL7689249 0.79 RAB9A (0.48) RAB9ANPC1SMN1; SMN2GAAPOLB
SCHEMBL7688380 0.78 RAB9A (0.76) RAB9ANPC1SMN1; SMN2GAAPOLB
SCHEMBL7686249 0.78 NPC1 (0.47) RAB9ANPC1SMN1; SMN2GAATP53
SCHEMBL7689730 0.75 RAB9A (0.51) RAB9ANPC1SMN1; SMN2GAAPOLB
SCHEMBL4062820 0.74 MGAM (0.51) GAAMGAMSIMGAM2TDP1
SCHEMBL4359045 0.73 MGAM (0.51) GAAMGAMSIMGAM2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255494-B1 SUBSTITUTED BENZIMIDAZOLES USEFUL IN TREATING OR PREVENTING CONDITIONS ASSOCIATED WITH EXCESS OF NEUROPEPTIDE Y (AROUND ARTERIES IN HEART, RESPIRATORY TRACT, GASTROINTESTINAL TRACT AND GENITOURINARY TRACT); ETIOLOGY OF PSYCHIATRIC DISORDERS ELI LILLY AND COMPANY 2001-07-03 US disclosed
EP-0871442-A1 BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1998-10-21 EP disclosed
WO-1997025041-A1 BENZIMIDZOLYL NEUROPEPTIDE Y RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed