SCHEMBL7965235

SCHEMBL7965235

COC(=O)c1cc(-c2cc(C)cnc2F)cnc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP46A1 Q9Y6A2 1/20 0.38
ATM Q13315 1/20 0.38
WDR5 P61964 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
GAA P10253 1/20 0.37
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37
RAB9A P51151 1/20 0.37
SENP8 Q96LD8 1/20 0.37
SENP7 Q9BQF6 1/20 0.37
SENP6 Q9GZR1 1/20 0.37
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
EIF2S1 P05198 1/20 0.36
EIF2AK3 Q9NZJ5 1/20 0.36
OPRK1 P41145 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1847871 0.87 WDR5 (0.38) CYP46A1ATMWDR5SMN1; SMN2NPC1
SCHEMBL12024798 0.81 ATM (0.50) CYP46A1ATMGAAKDM4EALDH1A1
SCHEMBL1854206 0.79 AXL (0.47) CYP46A1GAARAB9AKDM4EL3MBTL1
SCHEMBL3980095 0.75 OPRK1 (0.47) ATMSMN1; SMN2GAANPC1CASP3
SCHEMBL7093171 0.73 AXL (0.60) SMN1; SMN2GAAHPGDKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7093169 0.71 AXL (0.59) SMN1; SMN2GAAHPGDKDM4EALDH1A1
SCHEMBL401530 0.71 OPRK1 (0.47) CYP46A1ATMSMN1; SMN2GAANPC1
SCHEMBL25547252 0.71 GRIN2B (0.41) CYP46A1AXL
SCHEMBL645628 0.70 ATM (0.44) ATMSMN1; SMN2GAANPC1RAB9A
SCHEMBL38664726 0.70 CA12 (0.50) ATMGAAHPGDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010017260-A1 TRIPYRIDYL CARBOXAMIDE OREXIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2010-02-11 WO disclosed