SCHEMBL7965986

SCHEMBL7965986

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCN(C)CC2)ccc1C(=O)Nc1cccc2[nH]c(NCCN(C)C)nc12

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.34
AVPR2 P30518 3/20 0.34
AVPR1A P37288 3/20 0.34
AVPR1B P47901 2/20 0.34
MAP3K7 O43318 3/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
LCK P06239 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
IRAK4 Q9NWZ3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7967145 0.99 PTGES (0.34) PTGESAVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL7975663 0.97 PTGES (0.36) PTGESAVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL7978293 0.95 AVPR2 (0.34) PTGESAVPR2AVPR1AAVPR1BMAP3K7
Hydrochloric Acid SCHEMBL7963628 0.95 AVPR2 (0.34) PTGESAVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL7975620 0.94 AVPR2 (0.34) AVPR2AVPR1AAVPR1BMAP3K7LCK
Hydrochloric Acid SCHEMBL7953946 0.94 AVPR2 (0.34) AVPR2AVPR1AAVPR1BMAP3K7LCK
SCHEMBL7967127 0.94 AVPR2 (0.34) PTGESAVPR2AVPR1AAVPR1BMAP3K7
Hydrochloric Acid SCHEMBL7978209 0.93 AVPR2 (0.33) PTGESAVPR2AVPR1AAVPR1BMAP3K7
SCHEMBL7483272 0.93 AVPR2 (0.37) PTGESAVPR2AVPR1AAVPR1BMAP3K7
Hydrochloric Acid SCHEMBL7953655 0.93 AVPR2 (0.37) PTGESAVPR2AVPR1AAVPR1BMAP3K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed