SCHEMBL7966418

SCHEMBL7966418

Cc1cnccc1NC(=O)c1cn(C2CC2)c2ncccc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.44
KCNH2 Q12809 5/20 0.44
PDE4A P27815 4/20 0.43
ELANE P08246 1/20 0.40
IKBKE Q14164 2/20 0.40
TBK1 Q9UHD2 2/20 0.40
KDM4E B2RXH2 1/20 0.39
KDM6B O15054 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
TYK2 P29597 1/20 0.39
IRAK4 Q9NWZ3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966474 0.96 PKM (0.42) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7966470 0.96 PKM (0.42) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7951623 0.87 KCNH2 (0.37) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7951625 0.87 KCNH2 (0.37) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7966583 0.85 KCNH2 (0.49) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7960320 0.85 KCNH2 (0.49) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7960147 0.84 HTT (0.51) PKMKCNH2PDE4AELANEKDM4E
SCHEMBL7960497 0.83 CNR1 (0.51) PKMKCNH2PDE4AELANECNR1
SCHEMBL7960214 0.83 KCNH2 (0.49) PKMKCNH2PDE4AELANEIKBKE
SCHEMBL7168115 0.82 KCNH2 (0.58) KCNH2PDE4AIKBKETBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331548-B1 PREVENTION OR TREATMENT OF CYTOKINE RELATED DISEASES SUNTORY LIMITED (JP) 2001-12-18 US disclosed
EP-0978516-A1 1-CYCLOALKYL-1,8-NAPHTHYRIDIN-4-ONE DERIVATIVES WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SUNTORY LIMITED (JP) 2000-02-09 EP disclosed