SCHEMBL7966558

SCHEMBL7966558

CC(C)C(C#N)c1c(F)cccc1F

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ESR1 P03372 3/20 0.33
ESR2 Q92731 3/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
RIPK1 Q13546 1/20 0.33
DRD2 P14416 1/20 0.30
HTR2A P28223 1/20 0.30
HRH1 P35367 1/20 0.30
ACHE P22303 1/20 0.30
CUL4A Q13619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31126004 0.82 ESR1 (0.32) ESR1ESR2
SCHEMBL954647 0.78 ALDH1A1 (0.39) ALDH1A1GAACYP2C9CYP2C19CES2
SCHEMBL7956277 0.78 IDO1 (0.38) ALDH1A1GAACYP2C9ESR1ESR2
SCHEMBL31158379 0.73 ALDH1A1 (0.36) ALDH1A1GAACYP2C9CYP2C19CES2
SCHEMBL20534566 0.71 ALDH1A1 (0.51) ALDH1A1GAACYP2C9CYP2C19RIPK1
SCHEMBL19262108 0.70 CES2 (0.39) ALDH1A1CES2CES1DRD2HTR2A
SCHEMBL19716865 0.70 TSHR (0.46) ALDH1A1GAACYP2C9CYP2C19CES2
SCHEMBL6906077 0.70 TSHR (0.46) ALDH1A1GAACYP2C9CYP2C19CES2
SCHEMBL807528 0.69 TSHR (0.39) ALDH1A1GAACYP2C9CYP2C19CES2
SCHEMBL807556 0.69 CES2 (0.41) CES2CES1HTR2AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed