SCHEMBL7967267

SCHEMBL7967267

CNS(=O)(=O)c1cc(C(=O)CBr)ccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSTO1 P78417 1/20 0.53
POLB P06746 3/20 0.46
HSD17B10 Q99714 1/20 0.46
KDM4E B2RXH2 1/20 0.45
GSK3B P49841 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP1A2 P05177 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 2/20 0.43
HTT P42858 2/20 0.42
MAPK1 P28482 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA13 Q8N1Q1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13545186 0.87 GSTO1 (0.55) GSTO1POLBHSD17B10KDM4EL3MBTL1
SCHEMBL10962880 0.87 GSTO1 (0.62) GSTO1POLBHSD17B10KDM4EGSK3B
SCHEMBL11632341 0.86 POLB (0.42) GSTO1POLBHSD17B10KDM4EGSK3B
SCHEMBL11632049 0.86 POLB (0.44) GSTO1POLBHSD17B10KDM4EGSK3B
SCHEMBL11529122 0.86 POLB (0.45) POLBHSD17B10KDM4EGSK3BL3MBTL1
SCHEMBL11570844 0.84 GSTO1 (0.52) GSTO1POLBHSD17B10KDM4EL3MBTL1
SCHEMBL11630310 0.83 SMN1; SMN2 (0.45) GSTO1POLBHSD17B10KDM4EGSK3B
SCHEMBL11595726 0.83 F10 (0.46) GSTO1POLBHSD17B10KDM4EL3MBTL1
SCHEMBL11634252 0.83 SMN1; SMN2 (0.42) GSTO1POLBHSD17B10KDM4EGSK3B
SCHEMBL5511176 0.83 GSTO1 (0.51) GSTO1POLBHSD17B10KDM4EL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6172099-B1 CARBAZOLE, DIBENZOFURAN, OR DIBENZOTHIOPHENE DERIVATIVES; DIETETICS, ANTIDIABETIC AGENTS; ANTILIPEMICS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 2001-01-09 US disclosed
EP-0997458-A1 NOVEL TRICYCLIC COMPOUNDS HAVING SATURATED RINGS AND MEDICINAL COMPOSITIONS CONTAINING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 2000-05-03 EP disclosed
US-4156735-A SALIDIURETICS HOECHST AKTIENGESELLSCHAFT (DE) 1979-05-29 US disclosed
US-4129656-A Thiazolidine derivatives, salidiuretic compositions and methods of effecting salidiuresis employing them HOECHST AKTIENGESELLSCHAFT (DE) 1978-12-12 US disclosed
US-4125614-A DIURETIC HOECHST AKTIENGESELLSCHAFT (DE) 1978-11-14 US disclosed
US-4118501-A SALIDIURETIC ACTIVITY HOECHST AKTIENGESELLSCHAFT (DE) 1978-10-03 US disclosed
US-4061761-A Thiazolidine derivatives HOECHST AKTIENGESELLSCHAFT (DT) 1977-12-06 US disclosed