SCHEMBL7969129

SCHEMBL7969129

CC(C)C(C#N)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 4/20 0.43
ESR1 P03372 3/20 0.43
ESR2 Q92731 3/20 0.43
KIF11 P52732 1/20 0.41
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
DHODH Q02127 1/20 0.35
ACP3 P15309 1/20 0.35
FFAR1 O14842 3/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
ALDH1A1 P00352 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8425821 0.85 ESR1 (0.44) PDE2AESR1ESR2KIF11CES2
SCHEMBL18210542 0.80 PDE2A (0.46) PDE2AKIF11CES2CES1DHODH
SCHEMBL11824304 0.79 PNMT (0.45) ESR1ESR2CES2ACP3
SCHEMBL7967104 0.78 ESR1 (0.47) ESR1ESR2ALDH1A1
SCHEMBL4656621 0.77 PDE2A (0.43) PDE2AESR1ESR2KIF11CES2
SCHEMBL11444606 0.77 PDE2A (0.47) PDE2AESR1ESR2DHODHALDH1A1
SCHEMBL11157506 0.77 KDM4E (0.41) PDE2AESR1ESR2ALDH1A1
SCHEMBL17465918 0.75 KIF11 (0.47) PDE2AKIF11CES2CES1ACP3
SCHEMBL11161219 0.75 ESR1 (0.39) PDE2AESR1ESR2
SCHEMBL11445507 0.74 ESR1 (0.38) PDE2AESR1ESR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed