SCHEMBL7969465

SCHEMBL7969465

COc1ccc(CN2CCN(c3ncccn3)CC2)cc1-c1ccccc1

nearest known ligand 0.74

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.74
DRD4 P21917 5/20 0.74
DRD3 P35462 5/20 0.74
ALDH1A1 P00352 3/20 0.63
TSHR P16473 2/20 0.63
KDM4E B2RXH2 3/20 0.60
GAA P10253 1/20 0.60
HTR7 P34969 2/20 0.58
MAPK1 P28482 2/20 0.56
LMNA P02545 1/20 0.56
HTT P42858 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
PDE4B Q07343 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7959100 0.99 DRD2 (0.72) DRD2DRD4DRD3ALDH1A1TSHR
SCHEMBL7498064 0.85 DRD4 (1.00) DRD2DRD4DRD3ALDH1A1TSHR
SCHEMBL7958862 0.82 HTT (0.64) DRD2DRD4DRD3ALDH1A1KDM4E
SCHEMBL7972133 0.80 MEN1 (0.63) DRD2DRD4DRD3ALDH1A1TSHR
Maleic Acid SCHEMBL7991621 0.80 DRD4 (0.83) DRD2DRD4DRD3ALDH1A1TSHR
Fumaric Acid SCHEMBL7991623 0.80 DRD4 (0.83) DRD2DRD4DRD3ALDH1A1TSHR
Hydrochloric Acid SCHEMBL7968793 0.79 MEN1 (0.62) DRD2DRD4DRD3ALDH1A1TSHR
SCHEMBL3585542 0.78 ALDH1A1 (1.00) DRD2DRD4DRD3ALDH1A1TSHR
SCHEMBL7508845 0.76 DRD2 (1.00) DRD2DRD4DRD3ALDH1A1KDM4E
SCHEMBL8872544 0.76 ALDH1A1 (0.78) DRD2DRD4DRD3ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281359-B1 PSYCHOLOGICAL DISORDERS NEUROGEN CORPORATION 2001-08-28 US disclosed
US-6221871-B1 TREATING SCHIZOPHRENIA, DEPRESSION OR PARKINSON'S DISEASE NEUROGEN CORPORATION 2001-04-24 US disclosed
US-5912350-A Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands NEUROGEN CORPORATION (US) 1999-06-15 US disclosed
US-5594141-A ANTIPSYCHOTIC AND ANTIDEPRESSANT AGENTS; PARKINSON'S DISEASE NEUROGEN CORPORATION (US) 1997-01-14 US disclosed