SCHEMBL7969583

SCHEMBL7969583

CC/N=C(\NN)N1CCc2c(cnn2S(=O)(=O)c2ccc(C)cc2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.36
ALDH1A1 P00352 4/20 0.35
LMNA P02545 2/20 0.35
USP2 O75604 1/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 2/20 0.35
HSD17B10 Q99714 1/20 0.35
POLB P06746 2/20 0.35
PKM P14618 2/20 0.35
KDM2B Q8NHM5 1/20 0.34
KCNA1 Q09470 1/20 0.34
KCNAB1 Q14722 1/20 0.34
KMT2A Q03164 2/20 0.33
HTT P42858 1/20 0.33
NAMPT P43490 1/20 0.33
HTR6 P50406 1/20 0.33
HPGDS O60760 1/20 0.32
MAPT P10636 1/20 0.32
CD4 P01730 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1419569 1.00 NPSR1 (0.36) NPSR1ALDH1A1LMNAUSP2GAA
SCHEMBL1417531 0.83 ALDH1A1 (0.36) NPSR1ALDH1A1LMNAUSP2GAA
SCHEMBL1417529 0.83 ALDH1A1 (0.36) NPSR1ALDH1A1LMNAUSP2GAA
SCHEMBL1419555 0.81 KMT2A (0.37) NPSR1ALDH1A1LMNAUSP2GAA
SCHEMBL12677395 0.81 KMT2A (0.37) NPSR1ALDH1A1LMNAUSP2GAA
SCHEMBL12670985 0.77 KDM2B (0.38) ALDH1A1POLBPKMKDM2BKMT2A
SCHEMBL1417900 0.74 ESR2 (0.45) ALDH1A1LMNAUSP2GAASMN1; SMN2
SCHEMBL7985524 0.73 ALDH1A1 (0.39) ALDH1A1LMNAUSP2GAASMN1; SMN2
SCHEMBL12670982 0.73 ALDH1A1 (0.39) ALDH1A1LMNAUSP2GAASMN1; SMN2
SCHEMBL7987996 0.65 ALDH1A1 (0.39) NPSR1ALDH1A1LMNAUSP2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298747-A1 TRIAZOLE DERIVATIVE OR SALT THEREOF Astellas Pharma Inc. (JP) 2011-03-23 EP disclosed
WO-2010001946-A1 TRIAZOLE DERIVATIVE OR SALT THEREOF アステラス製薬株式会社 (JP) 2010-01-07 WO disclosed