SCHEMBL7969764

SCHEMBL7969764

Cc1ccc(C2CC(N(O)C(N)=O)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 3/20 0.47
ALDH1A1 P00352 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MAP1LC3B Q9GZQ8 1/20 0.36
FFAR1 O14842 1/20 0.36
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GRIN2B Q13224 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
KDM4E B2RXH2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969766 1.00 ALOX5 (0.47) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7972931 1.00 ALOX5 (0.47) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7973077 0.89 ALOX5 (0.40) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7973079 0.89 ALOX5 (0.40) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7972773 0.89 ALOX5 (0.40) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7972771 0.89 ALOX5 (0.40) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7972772 0.89 ALOX5 (0.40) ALOX5ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL7959777 0.83 ALOX5 (0.64) ALOX5ALDH1A1MAP1LC3BHTR2AHTR2C
SCHEMBL7972876 0.83 ALOX5 (0.47) ALOX5ALDH1A1HTR2CHTR2BNPC1
SCHEMBL7973196 0.83 ALOX5 (0.47) ALOX5ALDH1A1MAP1LC3BHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291520-B1 INHIBIT THE ENZYME LIPOXYGENASE; TREATMENT OR ALLEVIATION OF INFLAMMATORY DISEASES, ALLERGIC CONDITIONS AND CARDIOVASCULAR DISEASES PFIZER 2001-09-18 US disclosed
EP-0559743-B1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER (US) 1995-03-08 EP disclosed