SCHEMBL7969798

SCHEMBL7969798

CSc1nc2c(C(=O)O)cccc2[nH]1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 16/20 0.58
PARP1 P09874 2/20 0.57
KDM4E B2RXH2 1/20 0.56
HPGD P15428 1/20 0.56
ALDH1A1 P00352 1/20 0.49
TDP1 Q9NUW8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18786057 0.87 KDM4E (0.59) DHODHPARP1KDM4EHPGDALDH1A1
SCHEMBL6842031 0.86 PARP1 (0.66) DHODHPARP1
SCHEMBL15808958 0.84 PKN1 (0.62) DHODHPARP1KDM4EALDH1A1TDP1
SCHEMBL9725333 0.82 DHODH (0.77) DHODHPARP1KDM4EHPGD
SCHEMBL7475443 0.80 PARP1 (0.55) PARP1KDM4EHPGDALDH1A1TDP1
SCHEMBL1298127 0.79 PARP1 (0.73) DHODHPARP1KDM4EHPGD
SCHEMBL825449 0.78 KDM4E (0.73) DHODHPARP1KDM4EHPGD
SCHEMBL6519737 0.77 ALDH1A1 (0.42) DHODHPARP1KDM4EHPGDALDH1A1
Hydrochloric Acid SCHEMBL829317 0.77 KDM4E (0.71) DHODHPARP1KDM4EHPGD
SCHEMBL7863163 0.77 PARP1 (0.63) DHODHPARP1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6316482-B1 FOR THERAPY AND PROPHYLAXIS OF HYPERTENSION, HEART FAILURE, RENAL INSUFFICIENCY, EDEMA, ASCITES, VASOPRESSIN PARASECRETION SYNDROME, HEPATOCIRRHOSIS, HYPONATREMIA, HYPOKALEMIA, DIABETIC, CIRCULATION DISORDER, CEREBROVASCULAR DISEASE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-13 US disclosed
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed