SCHEMBL7969849

SCHEMBL7969849

NC(=O)N(O)C1C=C(c2ccccc2)C1

nearest known ligand 0.46

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.40
ALOX5 P09917 5/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9407414 0.73 ALOX5 (0.58) LMNAALOX5
SCHEMBL7969537 0.71 LMNA (0.37) LMNAALOX5
SCHEMBL27532209 0.71 ALOX5 (0.44) ALOX5
SCHEMBL9597226 0.68 ALOX5 (0.44) ALOX5
SCHEMBL7969806 0.67 ALOX5 (0.50) LMNAALOX5
Biphenyl SCHEMBL27435087 0.65 LMNA (0.48) LMNAALOX5
SCHEMBL7969404 0.64 ALOX5 (0.56) ALOX5
SCHEMBL7969402 0.64 ALOX5 (0.56) ALOX5
SCHEMBL7973050 0.64 ALOX5 (0.56) ALOX5
SCHEMBL16113017 0.64 AKR1C3 (0.40) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291520-B1 INHIBIT THE ENZYME LIPOXYGENASE; TREATMENT OR ALLEVIATION OF INFLAMMATORY DISEASES, ALLERGIC CONDITIONS AND CARDIOVASCULAR DISEASES PFIZER 2001-09-18 US disclosed
EP-0559743-B1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER (US) 1995-03-08 EP disclosed
EP-0559743-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE. PFIZER HOSPITAL PROD (US) 1993-09-15 EP disclosed
WO-1992009566-A1 NOVEL HYDROXAMIC ACID AND N-HYDROXYUREA DERIVATIVES AND THEIR USE PFIZER INC. (US) 1992-06-11 WO disclosed