SCHEMBL7970766

SCHEMBL7970766

[c]1ccc(C2CNCCCN2)cc1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
CHRNB2 P17787 2/20 0.32
CHRNA7 P36544 2/20 0.32
CHRNA4 P43681 2/20 0.32
MEN1 O00255 2/20 0.31
CYP2C19 P33261 2/20 0.31
KMT2A Q03164 2/20 0.31
POLB P06746 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2C9 P11712 1/20 0.31
HTR3A P46098 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16570136 0.89 CTSL (0.33)
SCHEMBL9829845 0.81 KDM1A (0.41) CYP2D6CHRNB2CHRNA7CHRNA4MEN1
SCHEMBL1030220 0.79 CHRNB2 (0.50) CYP2D6KCNH2CHRNB2CHRNA7CHRNA4
SCHEMBL1030421 0.79 CHRNB2 (0.50) CYP2D6KCNH2CHRNB2CHRNA7CHRNA4
SCHEMBL1031980 0.79 CHRNB2 (0.50) CYP2D6KCNH2CHRNB2CHRNA7CHRNA4
SCHEMBL6865588 0.78 CYP2D6 (0.37) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL28677309 0.78 SLC18A3 (0.42) CYP2D6CHRNB2CHRNA7CHRNA4MEN1
SCHEMBL6860743 0.78 CYP2D6 (0.37) CYP2D6SLC6A2SLC6A4SLC6A3KCNH2
SCHEMBL188416 0.77 MEN1 (0.51) CYP2D6CHRNB2CHRNA7CHRNA4MEN1
SCHEMBL27564375 0.77 MEN1 (0.51) CYP2D6CHRNB2CHRNA7CHRNA4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333320-B1 USEFUL AS DRUGS, ESPECIALLY AS AN ACTIVATED BLOOD COAGULATION FACTOR X INHIBITOR Yamanouchi Pharmaceutical Co. (JP) 2001-12-25 US disclosed
EP-1000936-A1 NOVEL HEXAHYDRO-1,4-DIAZEPINE DERIVATIVES OR SALTS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2000-05-17 EP disclosed