SCHEMBL7970844

SCHEMBL7970844

COC(=O)c1ccc2c(c1)/C(=C(/Nc1cccc(CN(C)C)c1)c1ccccc1)C(=O)N2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
HPGD P15428 1/20 0.44
RAB9A P51151 5/20 0.42
CASR P41180 1/20 0.42
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HSD17B10 Q99714 1/20 0.41
HIF1A Q16665 1/20 0.40
SENP1 Q9P0U3 1/20 0.40
PDPK1 O15530 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
AURKA O14965 1/20 0.39
RAF1 P04049 1/20 0.39
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
NPC1 O15118 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981209 0.91 PDPK1 (0.41) ALDH1A1HPGDRAB9AMEN1KMT2A
SCHEMBL6971260 0.90 JAK3 (0.41) ALDH1A1MEN1KMT2ASMN1; SMN2PDPK1
SCHEMBL6971265 0.90 JAK3 (0.41) ALDH1A1MEN1KMT2ASMN1; SMN2PDPK1
SCHEMBL6978475 0.89 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2AURKA
SCHEMBL6978482 0.89 MEN1 (0.40) ALDH1A1MEN1KMT2ASMN1; SMN2AURKA
SCHEMBL8189897 0.88 ALDH1A1 (0.48) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8189893 0.88 ALDH1A1 (0.48) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8191858 0.88 KIT (0.39) ALDH1A1HPGDRAB9AMEN1KMT2A
SCHEMBL8191861 0.88 KIT (0.39) ALDH1A1HPGDRAB9AMEN1KMT2A
SCHEMBL6982734 0.88 PPARG (0.39) ALDH1A1HPGDKMT2ASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed