SCHEMBL7971540

SCHEMBL7971540

CCn1c(-c2ccc(N)cc2)nnc1C(C)(C)Oc1c(F)cc(Cl)cc1F

nearest known ligand 0.76

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
ADRB2 P07550 1/20 0.34
APOBEC3A P31941 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPT P10636 2/20 0.33
HTT P42858 1/20 0.32
USP2 O75604 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984625 0.91 KDM4E (0.36) ALDH1A1KDM4EHPGDADRB2APOBEC3A
SCHEMBL7971805 0.91 KDM4E (0.36) ALDH1A1KDM4EHPGDADRB2APOBEC3A
SCHEMBL7992001 0.88 KDM4E (0.39) ALDH1A1KDM4EHPGDADRB2APOBEC3A
SCHEMBL7978690 0.87 HSD11B1 (0.36) KDM4E
SCHEMBL12671345 0.87 TSHR (0.40) ALDH1A1HPGDCYP2C9CYP2C19HTT
SCHEMBL7981464 0.87 KDM4E (0.36) ALDH1A1KDM4EHPGDADRB2APOBEC3A
SCHEMBL1417571 0.87 ALPG (0.38)
SCHEMBL1418321 0.85 DYRK1A (0.35)
SCHEMBL7984529 0.82 DYRK1A (0.35)
SCHEMBL7984651 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001946-A1 TRIAZOLE DERIVATIVE OR SALT THEREOF アステラス製薬株式会社 (JP) 2010-01-07 WO disclosed