SCHEMBL7971805

SCHEMBL7971805

CCn1c(-c2ccc(N)cc2)nnc1C(C)(C)Oc1c(F)cc(C)cc1F

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
ADRB2 P07550 1/20 0.35
APOBEC3A P31941 1/20 0.35
APOBEC3G Q9HC16 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984625 0.93 KDM4E (0.36) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL7971540 0.91 ALDH1A1 (0.37) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL7992001 0.90 KDM4E (0.39) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL12671412 0.87 CYP2C9 (0.36) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL7988236 0.86 JAK2 (0.39) KDM4EMAPT
SCHEMBL7982039 0.82 RORC (0.41) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL7985163 0.82 HSD11B1 (0.34)
SCHEMBL7979824 0.81 KDM4E (0.38) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL7981464 0.81 KDM4E (0.36) KDM4EALDH1A1HPGDADRB2APOBEC3A
SCHEMBL7982385 0.80 KIT (0.31) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010001946-A1 TRIAZOLE DERIVATIVE OR SALT THEREOF アステラス製薬株式会社 (JP) 2010-01-07 WO disclosed