SCHEMBL7971684

SCHEMBL7971684

CC(=O)c1ccc(-c2ccc(-c3nn(C)c(-c4nc5cc6c(cc5[nH]4)CNC6)c3O)cc2)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 1/20 0.40
CDK2 P24941 1/20 0.39
PRKCZ Q05513 1/20 0.39
CHEK2 O96017 5/20 0.36
BRD4 O60885 4/20 0.35
ATR Q13535 2/20 0.35
RHEB Q15382 1/20 0.35
F9 P00740 1/20 0.35
F10 P00742 1/20 0.35
F11 P03951 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PDE10A Q9Y233 1/20 0.34
HPSE Q9Y251 1/20 0.34
KDM1A O60341 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976222 0.91 CHEK2 (0.44) PRKCZCHEK2
SCHEMBL10139990 0.90 ATR (0.40) CDK2CHEK2ATRRHEBF9
SCHEMBL7975900 0.90 CHEK2 (0.40) CDK2CHEK2BRD4ATRRHEB
SCHEMBL7973155 0.89 F9 (0.39) NPBWR1CHEK2BRD4ATRF9
SCHEMBL7972135 0.88 PDE10A (0.37) CDK2CHEK2F9F10F11
SCHEMBL7970581 0.88 F9 (0.40) NPBWR1CHEK2BRD4ATRF9
SCHEMBL7970061 0.87 GUSB (0.39) CHEK2PDE10A
SCHEMBL7960814 0.87 NPC1 (0.39) BRD4RHEBPDE10A
SCHEMBL7970587 0.87 TOP1 (0.34) CHEK2ATRF9F10F11
SCHEMBL7971397 0.87 ALDH1A1 (0.39) NPBWR1CDK2PRKCZF9F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed