SCHEMBL7972632

SCHEMBL7972632

c1ccc2sc(NCCc3c[nH]cn3)nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.60
RAB9A P51151 5/20 0.60
MAPT P10636 2/20 0.55
ALDH1A1 P00352 1/20 0.55
LMNA P02545 1/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
QPCT Q16769 1/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
NPY1R P25929 7/20 0.45
GLS O94925 1/20 0.45
IDO1 P14902 1/20 0.44
KMT2A Q03164 3/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
MEN1 O00255 2/20 0.42
CASP3 P42574 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14394876 0.80 NPC1 (0.65) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL686607 0.78 ILK (0.42) NPC1RAB9AMAPTALDH1A1SMN1; SMN2
SCHEMBL686490 0.78 ILK (0.69)
SCHEMBL9358637 0.76 NPC1 (1.00) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL1981914 0.72 NPC1 (0.67) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL1664350 0.72 NPC1 (0.67) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL11207220 0.72 NPC1 (0.67) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL25057062 0.71 NPC1 (0.65) NPC1RAB9AMAPTALDH1A1LMNA
SCHEMBL8626317 0.71 NPC1 (0.65) NPC1RAB9AMAPTALDH1A1LMNA
Hydrochloric Acid SCHEMBL2124383 0.71 NPC1 (0.65) NPC1RAB9AMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE37303-E1 Imidazole compounds and their therapeutic applications INSTITUT NATIONAL DEL LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2001-07-31 US claimed
US-5708171-A HISTAMINE H3-RECEPTOR ANTAGONIST INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-01-13 US claimed
US-RE37303-E1 Imidazole compounds and their therapeutic applications INSTITUT NATIONAL DEL LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 2001-07-31 US disclosed
US-5747420-A HERBICIDES NIHON BAYER AGROCHEM K.K. (JP) 1998-05-05 US disclosed
US-5708171-A HISTAMINE H3-RECEPTOR ANTAGONIST INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-01-13 US disclosed
US-5559113-A ANTAGONISTS TO HISTAMINE H3 RECEPTORS, SEDATIVES, ANTICONVULSANTS, ANTIULCER AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE 1996-09-24 US disclosed
EP-0597088-A1 NOVEL IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC APPLICATIONS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1994-05-18 EP disclosed
WO-1993014070-A2 NOVEL IMIDAZOLE DERIVATIVES, THEIR PREPARATION AND THERAPEUTIC APPLICATIONS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1993-07-22 WO disclosed