SCHEMBL7972733

SCHEMBL7972733

Nc1ccc2c(c1)CC(Nc1ccccn1)C2

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
NOS2 P35228 1/20 0.40
ROCK1 Q13464 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39
PSENEN Q9NZ42 1/20 0.39
HRH4 Q9H3N8 1/20 0.39
GBA1 P04062 1/20 0.38
KDM5A P29375 1/20 0.38
NPC1 O15118 1/20 0.37
PKM P14618 1/20 0.37
RAB9A P51151 1/20 0.37
GRIN2B Q13224 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15594516 0.84 HDAC8 (0.50) HDAC8HDAC6NOS2ROCK1SMN1; SMN2
SCHEMBL7970294 0.83 HDAC8 (0.47) HDAC8HDAC6ROCK1SMN1; SMN2PSEN1
SCHEMBL30724682 0.82 HDAC8 (0.54) HDAC8HDAC6NOS2ROCK1HRH4
SCHEMBL24982439 0.80 NPC1 (0.46) NPC1PKMRAB9A
SCHEMBL22010868 0.80 NPC1 (0.46) NPC1PKMRAB9A
SCHEMBL6490792 0.77 GRM5 (0.54) HDAC8HDAC6PSEN1PSEN2APH1B
SCHEMBL4058385 0.76 PSEN1 (0.46) SMN1; SMN2PSEN1PSEN2APH1BNCSTN
SCHEMBL4392502 0.76 SMO (0.53) SMN1; SMN2GRIN2B
SCHEMBL7909108 0.76 SMO (0.53) SMN1; SMN2GRIN2B
SCHEMBL8208327 0.75 GBA1 (0.44) HRH4GBA1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001005767-A1 ORGANIC COMPOUNDS NOVARTIS AG (CH) 2001-01-25 WO claimed