SCHEMBL7972856

SCHEMBL7972856

C#CC(=O)C1CNCCN1NC(=O)c1ccc(F)cc1.c1cc2ccc1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.39
PTPN1 P18031 2/20 0.37
CD274 Q9NZQ7 1/20 0.36
FPR2 P25090 1/20 0.36
SCN9A Q15858 1/20 0.36
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
CTSC P53634 1/20 0.34
GPR6 P46095 1/20 0.34
HSD11B1 P28845 1/20 0.34
MCHR1 Q99705 1/20 0.34
CHRM4 P08173 1/20 0.34
BCL9 O00512 1/20 0.34
CTNNB1 P35222 1/20 0.34
WNT1 P04628 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972579 0.83 CYP2D6 (0.40) CYP2D6PTPN1CD274FPR2SCN9A
SCHEMBL8419841 0.81 CYP2D6 (0.47) CYP2D6GPR6HSD11B1
Water SCHEMBL7778613 0.80 CYP2D6 (0.46) CYP2D6CTSBCTSSCTSKCTSC
SCHEMBL7972859 0.73 HSD11B1 (0.49) CYP2D6HSD11B1
SCHEMBL1721295 0.68 CYP2D6 (0.67) CYP2D6GPR6
Bromide SCHEMBL7777483 0.67 CYP2D6 (0.65) CYP2D6GPR6
SCHEMBL28624849 0.63 HTT (0.45)
Bromide SCHEMBL7972483 0.63 CYP2D6 (0.58) CYP2D6GPR6
SCHEMBL9168347 0.62 SMN1; SMN2 (0.44)
SCHEMBL8587416 0.62 NPC1 (0.43) CYP2D6DRD2DRD4CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6291464-B1 POTENTIATION OF THE CHOLINERGIC ACTIVITY; THERAPEUTIC TREATMENT OF AMNESIA, DEMENTIA OR SENILE DEMENTIA FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-09-18 US disclosed