SCHEMBL7973532

SCHEMBL7973532

CCOC(=O)c1ccc(Oc2ccc(CC(C)(C)N)cc2)nc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.51
OPRM1 P35372 8/20 0.46
OPRD1 P41143 8/20 0.46
OPRK1 P41145 7/20 0.46
LMNA P02545 3/20 0.43
MAPT P10636 2/20 0.43
TSHR P16473 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
MAOA P21397 1/20 0.43
GRIN2D O15399 1/20 0.42
GRIN3B O60391 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A3 Q01959 1/20 0.42
GRIN1 Q05586 1/20 0.42
KCNH2 Q12809 1/20 0.42
GRIN2A Q12879 1/20 0.42
GRIN2B Q13224 1/20 0.42
ROCK1 Q13464 1/20 0.42
GRIN2C Q14957 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971486 0.88 LMNA (0.56) OPRM1OPRD1OPRK1LMNAGRIN2D
SCHEMBL20482160 0.86 PDE4B (0.57) PDE4BOPRM1OPRD1OPRK1LMNA
SCHEMBL3691973 0.85 OPRM1 (0.61) OPRM1OPRD1OPRK1GRIN2DGRIN3B
SCHEMBL5831347 0.85 LMNA (0.55) LMNAMAPTTSHRCYP1A2CYP3A4
SCHEMBL20482499 0.83 PDE4B (0.54) PDE4BOPRM1OPRD1OPRK1LMNA
SCHEMBL19362909 0.83 PDE4B (0.54) PDE4BLMNAMAPTTSHRNPSR1
SCHEMBL19362950 0.82 PDE4B (0.58) PDE4BLMNAMAPTTSHRKMT2A
SCHEMBL6179875 0.81 PDE4B (0.57) PDE4BOPRM1OPRD1OPRK1LMNA
SCHEMBL21656688 0.81 PDE4B (0.53) PDE4BOPRM1OPRD1OPRK1LMNA
SCHEMBL19363006 0.81 PDE4B (0.53) PDE4BLMNAMAPTTSHRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001036412-A1 PROCESS FOR THE PREPARATION OF ARYLOXY PROPANOLAMINES ELI LILLY AND COMPANY (US) 2001-05-25 WO disclosed