SCHEMBL7974371

SCHEMBL7974371

COc1c2c(c(OC)c(OC)c1OC)CC(CCCCCCCCN1C(=O)c3ccccc3C1=O)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.48
ALDH1A1 P00352 2/20 0.48
MEN1 O00255 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
ALOX12 P18054 1/20 0.48
ADRA1D P25100 1/20 0.48
HTR7 P34969 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
KMT2A Q03164 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KDM4E B2RXH2 1/20 0.47
GLA P06280 1/20 0.47
HPGD P15428 1/20 0.47
DRD2 P14416 2/20 0.47
DRD3 P35462 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974325 0.85 HTR1A (0.48) HTR1AALDH1A1MEN1CYP3A4CYP2D6
SCHEMBL7961134 0.76 HCAR2 (0.31)
SCHEMBL29263737 0.74 HPGD (0.59) HTR1AALDH1A1HTR7HPGDDRD3
SCHEMBL3476989 0.73 ACHE (0.81) HTR1AHTR7KMT2ADRD3CYP1A2
SCHEMBL14450985 0.73 ACHE (0.57) HTR1AALDH1A1HTR7HPGDDRD3
SCHEMBL31128445 0.72 HDAC8 (0.47) ALDH1A1MEN1KMT2AHSD17B10KDM4E
SCHEMBL8862878 0.72 TDP1 (0.75) MEN1KMT2ACYP1A2CYP2C19ACHE
SCHEMBL6777483 0.72 TDP1 (0.75) MEN1KMT2ACYP1A2CYP2C19ACHE
SCHEMBL8863154 0.72 TDP1 (0.75) MEN1KMT2ACYP1A2CYP2C19ACHE
SCHEMBL2604742 0.72 TDP1 (0.75) MEN1KMT2ACYP1A2CYP2C19ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6326369-B1 ALZHEIMER'S DISEASE TAKEDA CHEMICALS INDUSTRIES, LTD. (JP) 2001-12-04 US disclosed