SCHEMBL7975541

SCHEMBL7975541

c1ccc(COCc2cccc3[nH]c(-c4ccccc4)nc23)cc1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
GRIN2B Q13224 1/20 0.54
DHODH Q02127 7/20 0.52
PRMT5 O14744 2/20 0.48
PARP1 P09874 3/20 0.47
GAA P10253 7/20 0.46
MGAM O43451 6/20 0.46
SI P14410 6/20 0.46
MGAM2 Q2M2H8 6/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8816937 0.85 CYP1A2 (0.59) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL6687964 0.78 GRIN2B (0.60) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL3969183 0.78 GRIN2B (0.60) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL6686102 0.77 MGAM (0.62) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL7210788 0.75 GRIN2B (0.58) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL7211155 0.75 GRIN2B (0.58) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL30615069 0.72 MGAM (0.76) PARP1GAAMGAMSIMGAM2
SCHEMBL5074029 0.72 MGAM (0.76) PARP1GAAMGAMSIMGAM2
SCHEMBL8814837 0.72 GRIN2B (0.54) CYP1A2CYP2D6GRIN2BDHODHPARP1
SCHEMBL7461763 0.72 GRIN2B (0.54) CYP1A2CYP2D6GRIN2BDHODHPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194396-B1 ANTIALLERGENS; ANTIINFLAMMATION AGENTS; AUTOIMMUNE DISEASE; ANTISHOCK AGENTS; ANALGESICS; E.G., A 4 OR 7-PHENYLALKYLENE-OXYBENZIMIDAZOLE UNSUBSTITUTED OR SUBSTITUTED IN THE 1,2,3-POSITION WITH AN OXY, AMINO AND/OR THIO GROUP FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-02-27 US disclosed