SCHEMBL7976563

SCHEMBL7976563

N#Cc1ccc2c(c1)c(-c1cncc(-c3ccc(Cl)cc3)c1)cn2CCN1CCCCC1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.52
FLT1 P17948 3/20 0.47
FLT4 P35916 3/20 0.47
SCN7A Q01118 1/20 0.41
SLC6A4 P31645 1/20 0.39
HRH3 Q9Y5N1 7/20 0.38
SIGMAR1 Q99720 2/20 0.38
MCHR1 Q99705 5/20 0.38
CYP2D6 P10635 1/20 0.37
CHRM1 P11229 1/20 0.37
HTR2A P28223 1/20 0.37
HRH2 P25021 1/20 0.36
HRH1 P35367 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7548699 0.94 KDR (0.54) KDRFLT1FLT4SCN7ASLC6A4
SCHEMBL7990347 0.92 KDR (0.53) KDRFLT1FLT4SLC6A4HRH3
SCHEMBL7555484 0.90 KDR (0.59) KDRFLT1FLT4SCN7AHRH3
SCHEMBL7987947 0.90 KDR (0.52) KDRFLT1FLT4SCN7AHRH3
SCHEMBL7555601 0.89 KDR (0.58) KDRFLT1FLT4SIGMAR1MCHR1
SCHEMBL7987153 0.88 KDR (0.50) KDRFLT1FLT4SCN7AHRH3
SCHEMBL7553614 0.86 KDR (0.55) KDRFLT1FLT4SLC6A4MCHR1
SCHEMBL7555658 0.85 KDR (0.73) KDRFLT1FLT4SCN7ASIGMAR1
SCHEMBL7547180 0.85 KDR (0.60) KDRFLT1FLT4HRH3HRH2
SCHEMBL7552695 0.85 KDR (0.54) KDRFLT1FLT4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed