SCHEMBL7987153

SCHEMBL7987153

COc1ccc(-c2cncc(-c3cn(CCN4CCCCC4)c4ccc(C#N)cc34)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.50
FLT1 P17948 3/20 0.45
FLT4 P35916 3/20 0.45
KDM1A O60341 1/20 0.43
HRH3 Q9Y5N1 3/20 0.43
HRH2 P25021 1/20 0.41
HRH1 P35367 1/20 0.41
MCHR1 Q99705 1/20 0.41
SCN7A Q01118 2/20 0.39
CHRNB1 P11230 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNB3 Q05901 1/20 0.39
ESR1 P03372 2/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7554511 0.95 KDR (0.51) KDRFLT1FLT4KDM1AHRH3
SCHEMBL7504415 0.91 KDR (0.50) KDRFLT1FLT4KDM1AESR1
SCHEMBL7549155 0.90 KDR (0.56) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7976563 0.88 KDR (0.52) KDRFLT1FLT4HRH3HRH2
SCHEMBL7555484 0.88 KDR (0.59) KDRFLT1FLT4HRH3SCN7A
SCHEMBL7511178 0.88 KDR (0.54) KDRFLT1FLT4KDM1AHRH3
SCHEMBL7554609 0.86 KDR (0.52) KDRFLT1FLT4CHRNB1CHRNB2
SCHEMBL7556122 0.85 KDR (0.51) KDRFLT1FLT4HRH3ESR1
SCHEMBL7555221 0.85 KDR (0.68) KDRFLT1FLT4FLT3
SCHEMBL7554276 0.84 KDR (0.52) KDRFLT1FLT4MCHR1CHRNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed