SCHEMBL7976571

SCHEMBL7976571

Cn1cc(C2=C(c3cn(C)c4cc(N5CCOCC5)ccc34)C(=O)NC2=O)c2ccc(F)cc21

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 16/20 0.56
PRKCA P17252 6/20 0.54
CDK2 P24941 3/20 0.51
CCNE2 O96020 2/20 0.51
CDK4 P11802 2/20 0.51
CCND1 P24385 2/20 0.51
CCNE1 P24864 2/20 0.51
PRKACA P17612 1/20 0.51
PRKACG P22612 1/20 0.51
PRKACB P22694 1/20 0.51
PRKCB P05771 5/20 0.47
PRKCE Q02156 3/20 0.47
PRKCG P05129 6/20 0.47
PRKCD Q05655 1/20 0.46
CDK1 P06493 1/20 0.46
PRKCQ Q04759 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7598834 0.91 CDK4 (0.65) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7988158 0.91 GSK3B (0.51) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7977136 0.88 GSK3B (0.57) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7530443 0.88 GSK3B (0.72) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7976147 0.87 GSK3B (0.56) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7976579 0.87 GSK3B (0.56) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7987080 0.87 GSK3B (0.54) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7976484 0.85 GSK3B (0.54) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7526149 0.85 GSK3B (0.53) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL7976559 0.84 GSK3B (0.53) GSK3BPRKCACDK2CCNE2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US claimed
US-6281356-B1 ANTICANRCER AGENTS HOFFMANN-LA ROCHE INC. 2001-08-28 US disclosed