SCHEMBL7976884

SCHEMBL7976884

CNc1cc2c(Nc3cccc(Cl)c3)ncnc2cn1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 1.00
ERBB2 P04626 3/20 0.74
MEN1 O00255 3/20 0.74
KMT2A Q03164 3/20 0.74
MKNK1 Q9BUB5 2/20 0.74
TNK2 Q07912 1/20 0.74
FADS1 O60427 1/20 0.62
KDM4E B2RXH2 3/20 0.62
MAPT P10636 3/20 0.62
CYP1A2 P05177 2/20 0.62
CYP3A4 P08684 2/20 0.62
CYP2D6 P10635 2/20 0.62
NPC1 O15118 1/20 0.62
PRNP P04156 1/20 0.62
CYP2C9 P11712 1/20 0.62
CYP2C19 P33261 1/20 0.62
HTT P42858 1/20 0.62
MAPK1 P28482 2/20 0.61
FBP1 P09467 2/20 0.61
GMNN O75496 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7965274 0.86 EGFR (1.00) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL7978486 0.85 EGFR (1.00) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL14040743 0.85 EGFR (0.76) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL1262166 0.85 EGFR (1.00) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL7978403 0.82 EGFR (0.73) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL7978491 0.82 EGFR (1.00) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL8817803 0.81 EGFR (0.74) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL22604128 0.81 EGFR (0.67) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL8817814 0.80 EGFR (0.68) EGFRERBB2MEN1KMT2AMKNK1
SCHEMBL4355658 0.80 EGFR (1.00) EGFRERBB2MEN1KMT2AMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6313292-B1 REACTION FROM 5-AMINO-2-FLUOROPYRIDINE; AMINATION, CYCLIZATION, CHLORINATION, SALT FORMATION, DECHLORINATION, DEBLOCKING WARNER-LAMBERT COMPANY 2001-11-06 US claimed
WO-1997026259-A1 IMPROVED PROCESS FOR PREPARING 4,6-DISUBSTITUTED PYRIDO[3,4-d]PYRIMIDINES WARNER-LAMBERT COMPANY (US) 1997-07-24 WO claimed
US-6313292-B1 REACTION FROM 5-AMINO-2-FLUOROPYRIDINE; AMINATION, CYCLIZATION, CHLORINATION, SALT FORMATION, DECHLORINATION, DEBLOCKING WARNER-LAMBERT COMPANY 2001-11-06 US disclosed
WO-1997026259-A1 IMPROVED PROCESS FOR PREPARING 4,6-DISUBSTITUTED PYRIDO[3,4-d]PYRIMIDINES WARNER-LAMBERT COMPANY (US) 1997-07-24 WO disclosed