SCHEMBL7977309

SCHEMBL7977309

COC(=O)c1ccc(Oc2ccc(C(Cc3ccncc3)c3ccc(OC(F)F)c(OC(F)F)c3)cn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 19/20 0.52
KCNH2 Q12809 2/20 0.46
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987426 0.89 PDE4A (0.65) PDE4AKCNH2
SCHEMBL7976870 0.85 PDE4A (0.56) PDE4AKCNH2
SCHEMBL7379831 0.85 PDE4A (0.58) PDE4AKCNH2
SCHEMBL7384382 0.84 PDE4A (0.57) PDE4AKCNH2
SCHEMBL7383186 0.84 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7994385 0.83 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7977065 0.82 LMNA (0.51) PDE4ALMNA
SCHEMBL7994691 0.82 PDE4A (0.53) PDE4AKCNH2
SCHEMBL7392833 0.82 PDE4A (0.54) PDE4AKCNH2
SCHEMBL7991272 0.82 LMNA (0.50) PDE4ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US claimed
US-6180650-B1 ANTIINFLAMMATORY AGENTS; RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTITUMOR AGENTS MERCK FROSST CANADA & CO. (CA) 2001-01-30 US disclosed