SCHEMBL7989198

SCHEMBL7989198

COc1cc2c(cc1OCc1ccccc1)CCN=C2C(=O)c1ccccc1O

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
HPGD P15428 1/20 0.57
GLA P06280 1/20 0.49
RCE1 Q9Y256 1/20 0.49
RAD52 P43351 1/20 0.45
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CHRNA7 P36544 2/20 0.43
GPR84 Q9NQS5 1/20 0.43
CTSV O60911 1/20 0.41
CTSL P07711 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
GAA P10253 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7991324 0.92 KDM4E (0.56) KDM4EHPGDGLARCE1RAD52
SCHEMBL7988142 0.88 KDM4E (0.53) KDM4EHPGDGLARCE1RAD52
SCHEMBL7977247 0.88 KDM4E (0.52) KDM4EHPGDGLARCE1RAD52
SCHEMBL7991331 0.87 KDM4E (0.53) KDM4EHPGDGLARCE1RAD52
SCHEMBL7992415 0.85 KDM4E (0.51) KDM4EHPGDGLARCE1RAD52
SCHEMBL7987500 0.85 SMPD1 (0.53) KDM4EHPGDGLARCE1RAD52
SCHEMBL7977331 0.84 KDM4E (0.49) KDM4EHPGDGLARCE1RAD52
SCHEMBL7991437 0.83 KDM4E (0.48) KDM4EHPGDGLARCE1RAD52
SCHEMBL7991229 0.82 KDM4E (0.49) KDM4EHPGDGLARCE1RAD52
SCHEMBL7994703 0.80 KDM4E (0.45) KDM4EHPGDGLARCE1RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001055117-A1 NOVEL ISOQUINOLINE DERIVATIVES, PREPARATION METHOD AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES SERVIER (FR) 2001-08-02 WO disclosed