SCHEMBL7977490

SCHEMBL7977490

Cc1nc2c(c(-c3cccc(Cl)c3Cl)c1C(=O)OC(C)C)C(=O)CC(C)(C)C2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.55
CYP1A2 P05177 3/20 0.54
CYP2C9 P11712 3/20 0.54
CYP2C19 P33261 2/20 0.54
ALDH1A1 P00352 5/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CYP3A4 P08684 1/20 0.49
MAPK1 P28482 2/20 0.39
GSK3B P49841 1/20 0.39
NPSR1 Q6W5P4 2/20 0.37
ACHE P22303 2/20 0.37
CACNB4 O00305 1/20 0.37
CACNA1A O00555 1/20 0.37
CACNA1G O43497 1/20 0.37
CACNG3 O60359 1/20 0.37
CACNA1F O60840 1/20 0.37
CACNA1H O95180 1/20 0.37
BCHE P06276 1/20 0.37
CACNB3 P54284 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981878 0.89 LMNA (0.57) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL8802499 0.85 LMNA (0.44) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7977502 0.84 CYP1A2 (0.53) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7967602 0.81 CACNB4 (0.39) LMNAALDH1A1ACHECACNB4CACNA1A
SCHEMBL7981180 0.80 CACNB4 (0.38) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL8802939 0.80 LMNA (0.47) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL8804101 0.80 LMNA (0.46) LMNACYP1A2CYP2C9CYP2C19ALDH1A1
SCHEMBL7979243 0.74 CACNB4 (0.38) LMNAALDH1A1ACHECACNB4CACNA1A
SCHEMBL10748512 0.73 SMN1; SMN2 (0.42) LMNAALDH1A1MEN1KMT2ANPSR1
SCHEMBL7967452 0.73 CYP1A2 (0.55) LMNACYP1A2CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6194428-B1 BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 2001-02-27 US claimed
US-6194428-B1 BRAIN DISORDERS; PSYCHOLOGICAL DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 2001-02-27 US disclosed