SCHEMBL7977669

SCHEMBL7977669

Clc1ccc2c(c1)c(-c1cncc(-c3ccsc3)c1)cn2CCN1CCOCC1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.78
FLT1 P17948 5/20 0.78
FLT4 P35916 5/20 0.78
NFATC1 O95644 1/20 0.46
GSK3B P49841 1/20 0.46
DYRK1A Q13627 1/20 0.46
MAPT P10636 2/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
ATM Q13315 1/20 0.40
CYP2A6 P11509 1/20 0.40
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7993928 0.93 KDR (0.78) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7551421 0.91 KDR (0.77) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7976570 0.88 KDR (0.59) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7506453 0.87 KDR (1.00) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7991008 0.86 KDR (0.62) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7987864 0.86 KDR (0.74) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7505431 0.86 KDR (0.74) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7550302 0.86 KDR (0.78) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7976990 0.86 KDR (0.78) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7976915 0.86 KDR (0.59) KDRFLT1FLT4NFATC1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed