SCHEMBL7991008

SCHEMBL7991008

Clc1ccc2c(c1)c(-c1cncc(-c3ccccc3)c1)cn2CCN1CCOCC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.62
FLT1 P17948 3/20 0.62
FLT4 P35916 3/20 0.62
NFATC1 O95644 1/20 0.47
GSK3B P49841 1/20 0.47
DYRK1A Q13627 1/20 0.47
MAPT P10636 4/20 0.44
KDM4E B2RXH2 3/20 0.44
TSHR P16473 2/20 0.44
ALOX12 P18054 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
HTT P42858 2/20 0.43
TP53 P04637 1/20 0.43
MAPK1 P28482 1/20 0.43
ATM Q13315 1/20 0.43
ALDH1A1 P00352 2/20 0.42
SLC2A2 P11168 1/20 0.41
F2 P00734 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976570 0.94 KDR (0.59) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7976802 0.93 KDR (0.59) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7986691 0.92 KDR (0.62) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7555743 0.91 KDR (0.62) KDRFLT1FLT4HTTATM
SCHEMBL7548749 0.89 KDR (0.72) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7502516 0.88 KDR (0.77) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7990519 0.88 KDR (0.53) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7976794 0.87 KDR (0.53) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7987083 0.87 KDR (0.69) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7977669 0.86 KDR (0.78) KDRFLT1FLT4NFATC1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed