SCHEMBL7979642

SCHEMBL7979642

Cc1nc(-c2ccc(OCCCN3CCN(CC(N)C=O)CC3)cc2)no1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CXCR1 P25024 6/20 0.55
AOC3 Q16853 2/20 0.46
HRH3 Q9Y5N1 4/20 0.43
KCNH2 Q12809 2/20 0.43
HRH2 P25021 3/20 0.42
HRH1 P35367 3/20 0.42
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
NR1I2 O75469 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979630 0.83 HRH2 (0.62) CXCR1HRH3HRH2HRH1
SCHEMBL7243866 0.83 HRH2 (0.62) CXCR1HRH3HRH2HRH1
SCHEMBL7245509 0.80 CXCR1 (0.58) CXCR1AOC3HRH3KCNH2HRH2
SCHEMBL7979690 0.79 ATM (0.53) HRH3KCNH2HRH2HRH1RAB9A
SCHEMBL7254923 0.77 GPR119 (0.57) CXCR1HRH3HRH2HRH1
SCHEMBL7245375 0.77 HRH3 (0.58) HRH3HRH2HRH1
SCHEMBL26027547 0.74 ACACB (0.61) AOC3RAB9ANPC1NR1I2
SCHEMBL7301302 0.73 CXCR1 (0.69) CXCR1HRH3RAB9ANPC1MAPK1
SCHEMBL7294501 0.71 ACACB (0.69) AOC3RAB9ANPC1CA12CA1
SCHEMBL26022112 0.71 AOC3 (0.52) CXCR1AOC3RAB9ANPC1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001066534-A2 CYCLIC AND BICYCLIC DIAMINO HISTAMINE-3 RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2001-09-13 WO claimed