SCHEMBL7980096

SCHEMBL7980096

Cc1ncc(-c2cccc(NC(=NN)c3ccccc3F)c2)n1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 6/20 0.51
TP53 P04637 2/20 0.40
RGS12 O14924 2/20 0.38
PABPC1 P11940 1/20 0.38
MAPT P10636 1/20 0.37
POLB P06746 1/20 0.37
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
GSK3B P49841 4/20 0.37
FGFR3 P22607 4/20 0.37
KDR P35968 4/20 0.37
MAPK1 P28482 2/20 0.37
LCLAT1 Q6UWP7 1/20 0.37
ALDH1A1 P00352 1/20 0.36
FYN P06241 1/20 0.36
WNT1 P04628 1/20 0.36
CLK2 P49760 1/20 0.36
CLK3 P49761 1/20 0.36
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980094 1.00 DYRK1A (0.51) DYRK1ATP53RGS12PABPC1MAPT
SCHEMBL7128690 0.87 DYRK1A (0.40) DYRK1ATP53MAPTGAAGSK3B
SCHEMBL7128685 0.87 DYRK1A (0.40) DYRK1ATP53MAPTGAAGSK3B
SCHEMBL7117409 0.78 DYRK1A (0.41) DYRK1ATP53MAPTGAAGSK3B
SCHEMBL7117407 0.78 DYRK1A (0.41) DYRK1ATP53MAPTGAAGSK3B
SCHEMBL7984129 0.75 FGFR3 (0.42) DYRK1AGSK3BFGFR3KDRFYN
SCHEMBL7121296 0.75 CYP1A2 (0.50) DYRK1AGSK3BFGFR3KDRALDH1A1
Hydrochloric Acid SCHEMBL7123999 0.74 FGFR3 (0.41) DYRK1AGSK3BFGFR3KDRFYN
SCHEMBL7120271 0.73 DYRK1A (0.51) DYRK1ATP53RGS12PABPC1GAA
SCHEMBL7121293 0.73 FYN (0.40) DYRK1AGSK3BFGFR3KDRFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed