SCHEMBL7980936

SCHEMBL7980936

Bc1ccc(C(=O)OC)s1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.56
LMNA P02545 2/20 0.56
PPARG P37231 1/20 0.56
NCOA2 Q15596 1/20 0.56
NCOA1 Q15788 1/20 0.56
NCOA3 Q9Y6Q9 1/20 0.56
HPGD P15428 4/20 0.50
L3MBTL1 Q9Y468 3/20 0.50
TSHR P16473 3/20 0.50
MAPK1 P28482 2/20 0.50
ATM Q13315 1/20 0.50
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
MRGPRX4 Q96LA9 1/20 0.40
OPRD1 P41143 1/20 0.39
KDM4E B2RXH2 4/20 0.38
MAPT P10636 3/20 0.38
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70027 0.84 NPSR1 (0.67) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL25075387 0.79 NPSR1 (0.56) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL1303016 0.78 NPSR1 (0.60) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL1235256 0.78 LMNA (0.60) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL7902938 0.77 HPGD (0.38) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL425794 0.77 DAO (0.65) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL10671029 0.77 NPSR1 (0.58) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL277203 0.77 LMNA (0.58) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL8291932 0.76
SCHEMBL12319273 0.75 NPSR1 (0.56) NPSR1LMNAPPARGNCOA2NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011153319-A1 C-28 AMIDES OF MODIFIED C-3 BETULINIC ACID DERIVATIVES AS HIV MATURATION INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-12-08 WO disclosed
WO-2010009139-A2 IMIDAZOLYL PYRIMIDINE INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed
WO-2010009155-A2 FUSED HETEROCYCLYC INHIBITOR COMPOUNDS GILEAD COLORADO, INC. (US) 2010-01-21 WO disclosed
WO-2009137081-A2 SMALL MOLECULE INHIBITORS OF PLASMODIUM FALCIPARUM DIHYDROOROTATE DEHYDROGENASE MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2009-11-12 WO disclosed
EP-1807072-B1 CYCLOALKYL LACTAM DERIVATIVES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 LILLY CO ELI (US) 2009-01-07 EP disclosed