SCHEMBL7980994

SCHEMBL7980994

O=C1Nc2ccc(C(=O)O)cc2/C1=C(/Nc1ccc(CN2CCCCC2)cc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.48
HTT P42858 2/20 0.48
RAB9A P51151 2/20 0.48
HIF1A Q16665 2/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
LTA4H P09960 2/20 0.46
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
PDE5A O76074 1/20 0.43
ACHE P22303 1/20 0.43
HPGD P15428 1/20 0.43
TNIK Q9UKE5 1/20 0.43
EPAS1 Q99814 1/20 0.42
TNF P01375 1/20 0.42
LMNA P02545 2/20 0.42
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17976406 1.00 GAA (0.48) GAAHTTRAB9AHIF1ACYP2D6
SCHEMBL3149037 0.93 GAA (0.48) GAAHTTRAB9AHIF1ACYP2D6
SCHEMBL3149028 0.93 GAA (0.48) GAAHTTRAB9AHIF1ACYP2D6
SCHEMBL17976095 0.92 HIF1A (0.44) GAAHTTRAB9AHIF1ACYP2D6
SCHEMBL17976097 0.92 HIF1A (0.44) GAAHTTRAB9AHIF1ACYP2D6
SCHEMBL8192245 0.92 PRKAA2 (0.47) GAAHTTRAB9AALDH1A1KDM4E
SCHEMBL8192238 0.92 PRKAA2 (0.47) GAAHTTRAB9AALDH1A1KDM4E
SCHEMBL17976047 0.92 RET (0.49) RAB9AHIF1ALTA4HALDH1A1KDM4E
SCHEMBL17976049 0.92 RET (0.49) RAB9AHIF1ALTA4HALDH1A1KDM4E
SCHEMBL7982079 0.91 ALDH1A1 (0.51) GAAHTTRAB9ACYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
WO-2016131789-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-25 WO disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed
EP-3056202-A1 BENZOPYRROLIDONE DERIVATIVES POSSESSING ANTIVIRAL AND ANTICANCER PROPERTIES Max-Planck-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2016-08-17 EP disclosed
US-6169106-B1 ANTITUMOUR AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-01-02 US disclosed