SCHEMBL7981179

SCHEMBL7981179

CNc1nc(Cc2ccc(C(N)=NCC(=O)O)cc2)nc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.43
CYP1A2 P05177 4/20 0.42
CYP3A4 P08684 4/20 0.42
CLK4 Q9HAZ1 4/20 0.42
HSD17B10 Q99714 3/20 0.42
CYP2C9 P11712 2/20 0.42
USP2 O75604 2/20 0.42
TP53 P04637 1/20 0.42
BCHE P06276 1/20 0.42
PRNP P04156 2/20 0.41
RXFP1 Q9HBX9 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
CTNNB1 P35222 1/20 0.40
TCF7L2 Q9NQB0 1/20 0.40
PDE4B Q07343 1/20 0.39
L3MBTL1 Q9Y468 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7984282 0.70 MAPK1 (0.53) CYP1A2CYP3A4CLK4HSD17B10CYP2C9
SCHEMBL31649377 0.67 KDM4E (0.56) ACHECYP1A2CYP3A4CLK4HSD17B10
SCHEMBL3209937 0.66 PRNP (0.54) PRNPRXFP1NPSR1AURKAAURKB
SCHEMBL4859938 0.64 RAD52 (0.69) ACHEBCHENPSR1AURKAAURKB
SCHEMBL4866244 0.63 MAPK1 (0.59) ACHEBCHEKMT2AALDH1A1MAPK1
SCHEMBL13797204 0.62 CTNNB1 (0.86) CTNNB1TCF7L2
SCHEMBL16571758 0.62 MGAM (0.56) CYP1A2CYP2C9TP53PRNPRXFP1
SCHEMBL4864862 0.62 APP (0.68) ACHEBCHEL3MBTL1KMT2AMAPK1
SCHEMBL4532312 0.61 APP (0.67) CYP1A2CYP3A4CLK4HSD17B10CYP2C9
SCHEMBL13458341 0.61 KDM4E (0.59) ACHECYP1A2CYP3A4CLK4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6200976-B1 FOR TREATING THROMBOSIS BOEHRINGER INGELHEIM PHARMA KG (DE) 2001-03-13 US disclosed