SCHEMBL7981283

SCHEMBL7981283

Cc1cncc2c(C)c3cnccc3cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.43
MAOA P21397 2/20 0.42
KDM4E B2RXH2 3/20 0.41
HTT P42858 2/20 0.41
POLB P06746 2/20 0.41
RAD52 P43351 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.38
ACHE P22303 1/20 0.36
HASPIN Q8TF76 3/20 0.35
HIPK2 Q9H2X6 2/20 0.35
GRM4 Q14833 1/20 0.35
KIT P10721 3/20 0.34
ADORA3 P0DMS8 2/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
GMNN O75496 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
NR3C1 P04150 1/20 0.34
TP53 P04637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27109662 0.79 TOP2A (0.47) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL30656996 0.79 KDM4E (0.41) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL10200876 0.79 KDM4E (0.41) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL17051668 0.76 MAOA (0.45) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL10072720 0.74 TOP2A (0.55) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL10200877 0.73 KDM4E (0.42) KDM4EHTTNCOA3ACHEHIPK2
SCHEMBL3701838 0.72 CYP1A2 (0.52) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL2501659 0.72 TOP2A (0.45) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL21297740 0.71 KDM4E (0.47) TOP2AMAOAKDM4EHTTPOLB
SCHEMBL8404561 0.71 CYP2A6 (0.52) TOP2AMAOAKDM4EHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5994365-A BACTERICIDES; FUNGICIDES; ANTITUMOR AGENT DIAZANS LIMITED (CA) 1999-11-30 US claimed
WO-2001017997-A1 SUBSTITUTED DIAZAANTHRACENE COMPOUNDS HAVING PHARMACEUTICAL UTILITY DIAZANS LIMITED (CA) 2001-03-15 WO disclosed
US-5994365-A BACTERICIDES; FUNGICIDES; ANTITUMOR AGENT DIAZANS LIMITED (CA) 1999-11-30 US disclosed