SCHEMBL798137

SCHEMBL798137

O=C(NN1CCN(c2nc([AsH2])nc3sc(-c4cccnc4)nc23)CC1)c1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 4/20 0.48
CYP3A4 P08684 4/20 0.48
KCNH2 Q12809 3/20 0.48
LMNA P02545 2/20 0.40
CYP2D6 P10635 1/20 0.40
PTGS2 P35354 1/20 0.38
CYP1A2 P05177 2/20 0.38
CYP2C19 P33261 1/20 0.38
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CYP11B2 P19099 2/20 0.37
CYP11B1 P15538 1/20 0.37
DYRK1A Q13627 2/20 0.36
MAPT P10636 2/20 0.36
F2 P00734 1/20 0.36
ABL1 P00519 1/20 0.36
PDGFRB P09619 1/20 0.36
BCR P11274 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL654709 0.91 PI4KB (0.59) PI4KBCYP3A4KCNH2LMNACYP2D6
SCHEMBL798314 0.76 PI4KB (0.67) PI4KBCYP3A4KCNH2LMNAKMT2A
SCHEMBL655854 0.70 PI4KB (0.85) PI4KBCYP3A4KCNH2LMNACYP2C19
SCHEMBL1694319 0.69 PI4KB (0.60) PI4KBCYP3A4KCNH2LMNACYP2D6
SCHEMBL16650147 0.69 PI4KB (0.71) PI4KBCYP3A4KCNH2LMNACYP1A2
SCHEMBL655695 0.67 PI4KB (0.81) PI4KBCYP3A4KCNH2KMT2AMEN1
SCHEMBL15124766 0.67 PI4KB (0.56) PI4KBCYP3A4KCNH2LMNAPTGS2
SCHEMBL655530 0.67 PI4KB (0.85) PI4KBCYP3A4KCNH2PDGFRB
SCHEMBL655275 0.65 PI4KB (1.00) PI4KBCYP3A4KCNH2ALDH1A1SMN1; SMN2
SCHEMBL655972 0.65 PI4KB (0.69) PI4KBCYP3A4KCNH2SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP claimed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO claimed