SCHEMBL798314

SCHEMBL798314

O=C(Nc1ccc(C(F)(F)F)cc1)N1CCN(c2nc([AsH2])nc3sc(-c4cccnc4)nc23)CC1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PI4KB Q9UBF8 5/20 0.67
KCNH2 Q12809 3/20 0.67
CYP3A4 P08684 2/20 0.67
TRPV1 Q8NER1 8/20 0.58
MAPT P10636 2/20 0.50
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
KIT P10721 2/20 0.47
LMNA P02545 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL655695 0.91 PI4KB (0.81) PI4KBKCNH2CYP3A4TRPV1MAPT
SCHEMBL655530 0.80 PI4KB (0.85) PI4KBKCNH2CYP3A4KIT
SCHEMBL656344 0.80 PI4KB (0.84) PI4KBKCNH2CYP3A4TRPV1KMT2A
SCHEMBL655275 0.80 PI4KB (1.00) PI4KBKCNH2CYP3A4MAPTKIT
SCHEMBL651916 0.78 PI4KB (0.81) PI4KBKCNH2CYP3A4KIT
SCHEMBL798137 0.76 PI4KB (0.48) PI4KBKCNH2CYP3A4MAPTKMT2A
SCHEMBL654265 0.75 PI4KB (0.83) PI4KBKCNH2CYP3A4KIT
SCHEMBL1694319 0.73 PI4KB (0.60) PI4KBKCNH2CYP3A4TRPV1MAPT
SCHEMBL16650147 0.71 PI4KB (0.71) PI4KBKCNH2CYP3A4KITLMNA
SCHEMBL654793 0.70 PI4KB (0.81) PI4KBKCNH2CYP3A4MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2616077-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2013-07-24 EP disclosed
WO-2012035423-A1 ANTI-CANCER ACTIVITY OF NOVEL BICYCLIC HETEROCYCLES KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2012-03-22 WO disclosed