SCHEMBL798178

SCHEMBL798178

CCOC(=O)N(CC)c1ccc(F)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.49
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
POLQ O75417 3/20 0.42
HTT P42858 1/20 0.41
KMT2A Q03164 2/20 0.40
PTGIR P43119 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL798625 0.89 TSHR (0.49) TSHRALDH1A1CYP3A4SMN1; SMN2HTT
SCHEMBL28802321 0.87 TSHR (0.52) TSHRALDH1A1CYP3A4HTTKMT2A
SCHEMBL27901771 0.87 TSHR (0.49) TSHRALDH1A1CYP3A4SMN1; SMN2HTT
SCHEMBL9302078 0.82 ALDH1A1 (0.48) TSHRALDH1A1CYP3A4SMN1; SMN2NPC1
SCHEMBL31453537 0.82 MAPT (0.43) TSHRALDH1A1CYP3A4SMN1; SMN2NPC1
SCHEMBL8628786 0.80 ALDH1A1 (0.40) TSHRALDH1A1CYP3A4SMN1; SMN2NPC1
SCHEMBL8627774 0.80 ALDH1A1 (0.40) TSHRALDH1A1CYP3A4SMN1; SMN2NPC1
SCHEMBL5705196 0.79 TSHR (0.46) TSHRALDH1A1CYP3A4NPC1HTT
SCHEMBL29276174 0.78 TSHR (0.44) TSHRALDH1A1CYP3A4NPC1HTT
SCHEMBL9224528 0.77 TSHR (0.50) TSHRALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed