SCHEMBL7982291

SCHEMBL7982291

Cc1cc2c(cc1C)OC(C)C(=S)N2

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.33
BRD4 O60885 1/20 0.31
CREBBP Q92793 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971002 0.79 BRD4 (0.39) PARP1BRD4CREBBP
SCHEMBL7988135 0.79 BRD4 (0.53) PARP1BRD4CREBBP
SCHEMBL5671394 0.78 PARP1 (0.56) PARP1BRD4CREBBP
SCHEMBL7001562 0.77 MAPK9 (0.33) PARP1
SCHEMBL7144708 0.76 PDE3B (0.31)
SCHEMBL7711230 0.74 PARP1 (0.37) PARP1BRD4CREBBP
SCHEMBL7000943 0.74 PARP1 (0.37) PARP1BRD4CREBBP
SCHEMBL7000985 0.70 KDM4E (0.54) PARP1
SCHEMBL7981061 0.68 CREBBP (0.53) PARP1BRD4CREBBP
SCHEMBL7985936 0.68 PARP1 (0.38) PARP1BRD4CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6191127-B1 ANTIINFLAMMATORY AGENTS, AUTOIMMUNE DISEASES, CARDIOVASCULAR DISORDERS, NERVOUS SYSTEM DISORDERS SCHERING AKTIENGESELLSCHAFT (DE) 2001-02-20 US disclosed