SCHEMBL7982628

SCHEMBL7982628

CC(=O)SCCc1cn2cc(N)ccc2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.39
ABL1 P00519 1/20 0.39
RIN1 Q13671 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 5/20 0.39
ALDH1A1 P00352 4/20 0.39
POLB P06746 2/20 0.39
APP P05067 3/20 0.38
TP53 P04637 1/20 0.38
MCHR1 Q99705 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
RXFP1 Q9HBX9 1/20 0.34
METTL3 Q86U44 2/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
KLKB1 P03952 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969549 0.81 KDM4E (0.51) CYP2C19KDM4EALDH1A1TP53NPC1
SCHEMBL7986519 0.77 APP (0.38) CYP2C19KDM4EALDH1A1POLBAPP
SCHEMBL7980201 0.76 RAB9A (0.38) TDP1ABL1KDM4EALDH1A1POLB
SCHEMBL7982608 0.75 SMN1; SMN2 (0.45) KDM4EALDH1A1TP53NPC1RAB9A
SCHEMBL7969572 0.74 HRH4 (0.42) TDP1KDM4EALDH1A1POLBL3MBTL1
SCHEMBL31210804 0.74 APP (0.43) TDP1CYP2C19KDM4EALDH1A1POLB
SCHEMBL7979633 0.72 ERCC5 (0.34) CYP2C19KDM4EPOLBKLKB1MAPT
SCHEMBL20986013 0.72 APP (0.39) TDP1ABL1RIN1CYP2C19KDM4E
SCHEMBL7982714 0.71 KDM4E (0.44) TDP1KDM4EALDH1A1POLBL3MBTL1
SCHEMBL18883283 0.71 HRH4 (0.40) KDM4EALDH1A1POLBAPPNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed