SCHEMBL7982608

SCHEMBL7982608

CC(=O)SCCc1cn2cccc(N)c2n1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.45
MAPT P10636 3/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
DHFR P00374 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 5/20 0.38
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HSD17B10 Q99714 4/20 0.37
HPGD P15428 2/20 0.37
MAPK1 P28482 3/20 0.35
ADORA2A P29274 1/20 0.35
TP53 P04637 1/20 0.35
SIRT5 Q9NXA8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982677 0.78 SMN1; SMN2 (0.47) SMN1; SMN2MAPTNPC1RAB9ADHFR
SCHEMBL7969549 0.77 KDM4E (0.51) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL7982628 0.75 TDP1 (0.39) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL9226257 0.74 SMN1; SMN2 (0.52) SMN1; SMN2MAPTNPC1RAB9ADHFR
SCHEMBL7969399 0.74 ALDH1A1 (0.50) SMN1; SMN2MAPTNPC1RAB9ANPSR1
SCHEMBL7982689 0.72 ALDH1A1 (0.46) SMN1; SMN2MAPTNPC1RAB9ADHFR
SCHEMBL2489626 0.71 RAB9A (0.49) SMN1; SMN2MAPTNPC1RAB9ADHFR
SCHEMBL7980749 0.70 NOS2 (0.42) NPSR1
SCHEMBL7980201 0.70 RAB9A (0.38) SMN1; SMN2MAPTNPC1RAB9AALDH1A1
SCHEMBL7969572 0.68 HRH4 (0.42) SMN1; SMN2MAPTALDH1A1KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed