SCHEMBL7982689

SCHEMBL7982689

CCOC(=O)Cc1cn2cccc(N)c2n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
CHEK1 O14757 1/20 0.45
KDM4E B2RXH2 9/20 0.42
HSD17B10 Q99714 5/20 0.42
POLB P06746 3/20 0.42
THRB P10828 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX15 P16050 1/20 0.42
FPR1 P21462 1/20 0.42
CYP2C19 P33261 1/20 0.42
RECQL P46063 1/20 0.42
DHFR P00374 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20596629 0.86 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTLMNANPC1
SCHEMBL118201 0.79 ALDH1A1 (0.56) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL1668064 0.77 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2MAPTLMNANPC1
SCHEMBL9226257 0.77 SMN1; SMN2 (0.52) ALDH1A1SMN1; SMN2MAPTLMNANPC1
SCHEMBL20596644 0.76 KDM4E (0.41) ALDH1A1SMN1; SMN2MAPTLMNARAB9A
SCHEMBL20595996 0.74 KDM4E (0.43) ALDH1A1SMN1; SMN2MAPTLMNARAB9A
SCHEMBL20596557 0.74 MAPT (0.43) ALDH1A1SMN1; SMN2MAPTLMNARAB9A
SCHEMBL7982714 0.74 KDM4E (0.44) ALDH1A1SMN1; SMN2MAPTCHEK1KDM4E
SCHEMBL7986876 0.74 ALDH1A1 (0.64) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL2489626 0.74 RAB9A (0.49) ALDH1A1SMN1; SMN2MAPTLMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed