SCHEMBL7983595

SCHEMBL7983595

CCCC(=O)Oc1cn2ncccc2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 5/20 0.39
ALOX15 P16050 1/20 0.36
KMT2A Q03164 2/20 0.35
RAB9A P51151 2/20 0.35
BCL9 O00512 1/20 0.35
CTNNB1 P35222 1/20 0.35
PDE4B Q07343 4/20 0.33
PDE4C Q08493 4/20 0.33
PDE4D Q08499 4/20 0.33
PDGFRB P09619 1/20 0.33
PDGFRA P16234 1/20 0.33
GAA P10253 3/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GLA P06280 1/20 0.33
MAPT P10636 1/20 0.32
CA2 P00918 2/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
ELANE P08246 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982679 0.78 GAA (0.39) ALOX15KMT2ARAB9ABCL9CTNNB1
SCHEMBL7980862 0.78 PTGS1 (0.47) KMT2ARAB9AKDM4EALDH1A1MAPT
SCHEMBL2066827 0.74 PDE4A (0.38) PDE4ARAB9AGAAKDM4EALDH1A1
SCHEMBL7980755 0.73 MAPT (0.36) ALOX15KMT2ARAB9ABCL9CTNNB1
SCHEMBL7982712 0.71 BCL9 (0.34) ALOX15KMT2ARAB9ABCL9CTNNB1
SCHEMBL7981083 0.71 HRH4 (0.42) ALOX15KMT2ARAB9ABCL9CTNNB1
SCHEMBL7983599 0.69 PDE4A (0.47) PDE4AALOX15KMT2AGAAKDM4E
SCHEMBL17492364 0.69 GAA (0.62) PDE4AKMT2ARAB9AGAAKDM4E
SCHEMBL7986875 0.69 KDM4E (0.53) KMT2ARAB9AGAAKDM4EALDH1A1
SCHEMBL700968 0.68 PDE4A (0.45) PDE4AALOX15KMT2ARAB9ABCL9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed