SCHEMBL7986875

SCHEMBL7986875

CCCC(=O)Oc1cn2cccnc2n1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.53
ALDH1A1 P00352 9/20 0.53
HPGD P15428 7/20 0.53
RAB9A P51151 7/20 0.50
GLA P06280 7/20 0.47
GAA P10253 7/20 0.47
PDE5A O76074 1/20 0.46
HSD17B10 Q99714 5/20 0.46
CYP1A2 P05177 4/20 0.46
TP53 P04637 3/20 0.41
CYP2C9 P11712 2/20 0.41
MEN1 O00255 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
POLB P06746 4/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980862 0.77 PTGS1 (0.47) KDM4EALDH1A1HPGDRAB9AHSD17B10
SCHEMBL7982687 0.74 DHFR (0.41) KDM4EALDH1A1RAB9AHSD17B10MEN1
SCHEMBL7981083 0.73 HRH4 (0.42) KDM4EALDH1A1HPGDRAB9AGAA
SCHEMBL25347598 0.73 ALDH1A1 (0.56) KDM4EALDH1A1HPGDRAB9AGLA
SCHEMBL7986876 0.70 ALDH1A1 (0.64) KDM4EALDH1A1HPGDRAB9AGLA
SCHEMBL700968 0.70 PDE4A (0.45) KDM4EALDH1A1RAB9ACYP1A2TP53
SCHEMBL1407731 0.69 KDM4E (1.00) KDM4EALDH1A1HPGDRAB9AGLA
SCHEMBL9737854 0.69 ALDH1A1 (0.43) KDM4EALDH1A1RAB9AGLAGAA
SCHEMBL7983595 0.69 PDE4A (0.39) KDM4EALDH1A1RAB9AGLAGAA
SCHEMBL10205883 0.68 KDM4E (0.50) KDM4EALDH1A1HPGDRAB9AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed