SCHEMBL7981083

SCHEMBL7981083

CCCC(=O)Oc1cn2ccncc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.42
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
CLK1 P49759 1/20 0.37
DYRK1A Q13627 1/20 0.37
KDM4E B2RXH2 3/20 0.34
HPGD P15428 3/20 0.34
ALDH1A1 P00352 3/20 0.34
GAA P10253 2/20 0.34
CASP1 P29466 2/20 0.34
CASP7 P55210 2/20 0.34
HSD17B10 Q99714 2/20 0.34
ALOX15 P16050 2/20 0.34
ROCK1 Q13464 1/20 0.33
KMT2A Q03164 2/20 0.32
RAB9A P51151 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
BCL9 O00512 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980862 0.80 PTGS1 (0.47) KDM4EHPGDALDH1A1HSD17B10KMT2A
SCHEMBL7986875 0.73 KDM4E (0.53) KDM4EHPGDALDH1A1GAAHSD17B10
SCHEMBL7982712 0.73 BCL9 (0.34) KDM4EHPGDALDH1A1GAAALOX15
SCHEMBL3524087 0.73 PDE3B (0.45) HRH4PDE3BPDE3ACLK1DYRK1A
SCHEMBL7983595 0.71 PDE4A (0.39) KDM4EALDH1A1GAAALOX15KMT2A
SCHEMBL7981086 0.70 KDM4E (0.44) HRH4KDM4EHPGDALDH1A1GAA
SCHEMBL19997261 0.70 HRH4 (0.57) HRH4PDE3BPDE3ACLK1DYRK1A
SCHEMBL2922016 0.69 KDM4E (0.63) HRH4KDM4EHPGDALDH1A1GAA
SCHEMBL7986358 0.69 BCL9 (0.54) HPGDALDH1A1GAAKMT2ARAB9A
SCHEMBL25139484 0.69 HRH4 (0.52) HRH4PDE3BPDE3ACLK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed