SCHEMBL7983946

SCHEMBL7983946

OC1CCN(CCCc2ccccc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.70
CCR3 P51677 1/20 0.62
MEN1 O00255 1/20 0.62
TP53 P04637 1/20 0.62
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
TSHR P16473 1/20 0.62
CYP2C19 P33261 1/20 0.62
KMT2A Q03164 1/20 0.62
HTR2A P28223 1/20 0.60
KCNH2 Q12809 1/20 0.60
POLB P06746 1/20 0.60
SPHK1 Q9NYA1 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10438853 0.95 SIGMAR1 (0.69) SIGMAR1CCR3MEN1TP53CYP1A2
SCHEMBL9906601 0.91 SIGMAR1 (0.61) SIGMAR1CCR3MEN1TP53CYP1A2
SCHEMBL18922663 0.90 SIGMAR1 (0.61) SIGMAR1CCR3MEN1TP53CYP1A2
SCHEMBL4255190 0.89 ACHE (0.69) SIGMAR1CCR3CYP1A2CYP3A4CYP2D6
SCHEMBL4688942 0.85 SPHK1 (0.61) SIGMAR1SPHK1
SCHEMBL10522891 0.84 SIGMAR1 (0.72) SIGMAR1CCR3MEN1TP53CYP1A2
SCHEMBL3958257 0.84 HRH3 (0.58) SIGMAR1CCR3MEN1TP53CYP1A2
SCHEMBL7550067 0.83 SPHK1 (0.60) CYP1A2CYP3A4CYP2D6HTR2ASPHK1
SCHEMBL15650736 0.83 SIGMAR1 (0.60) SIGMAR1HTR2ASPHK1
SCHEMBL3452363 0.83 SPHK1 (0.60) SIGMAR1CCR3MEN1TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265434-B1 ANTIINFLAMMATORY AGENTS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000076511-A1 CYCLOPENTYL MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-12-21 WO disclosed
US-4886813-A INHIBITORS OF ANGIOTENSIN CONVERTING ENZYME OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 1989-12-12 US disclosed